From Chemistry to Biology, Medicine
and Material Science
 
  

 
 

 

THURSDAY, OCTOBER 15, 2009

 

13:30-14:45       Registration

 

1st Session

                        Chairs: Prof. Ioannis Gallos (Aristotle University of Thessaloniki)

                                    Assoc. Prof. Panagiota Minakakis (University of Athens)

                                               

14:45-15:00       Opening Remarks

15:00-15:45      Copper and Iridium Catalyzed Asymmetric Allylic Substitution

                        Prof. Alexandre Alexakis (University of Geneva, Switzerland)

15:45-16:10       Biomimetic Synthesis of Acremine G and Allomicrophyllone

                        Assoc. Prof.  Manolis Stratakis (University of Crete, Greece)

16:10-16:35       A Previleged Benzopyran Research and Development of New Synthetic Routes

                        Dr. Gerasimos Rassias (GlaxoSmithKline, UK)

16:35-16:55       Advances in Enantioselective Organocatalysis: Applications of Linchpin Catalysis

                        Dr. Christoforos G. Kokotos (Princeton University, USA)

16:55-17:30       Coffee Break

 

 

2nd Session

                        Chairs: Prof. Michael Orfanopoulos (University of Crete)

                                   Prof. Paul Cordopatis (University of Patras)

                                               

17:30-18:15       Carbon-Fluorine Bond: Construction and Deconstruction

                        Prof. Veronique Gouverneur (University of Oxford, UK)

18:15-18:40       The biodiversity in nature provides solutions to Synthetic Organic Chemists

                        Assoc. Prof. Thomas Mavromoustakos (University of Athens, Greece)

18:40-19:00       Looking for potent inhibitors of glycogen phosphorylase- the structure-based ligand design approach in vitro & in silico

                        Dr. Evaggelia D. Chrysina (National Hellenic Research Foundation, Greece)

19:00-19:20       Novel spirocyclic aminocyclitols: Simplified, rigid structures with antibiotic activity

                        Dr. Ioannis A. Katsoulis (N.C.S.R. “Demokritos”, Greece)

19:20                Cocktail

 

 

FRIDAY, OCTOBER 16, 2009

 

3rd Session

                        Chairs: Prof. Violetta Constantinou (Agricultural University of Athens)

                                   Prof. Nicholaos Ferderigos (University of Athens)

 

09:10-09:55      From Homer to Hedgehog: Synthesis of Cyclopamine Using a Biomimetic and Diastereoselective Approach

                        Prof. Athanassios Giannis (University of Leipzig, Germany

09:55-10:20      From Academic Research to its Exploitation for Medicinal Uses: Sartans, a New Generation of Drugs for Treating Hypertension and Cardiovascular Diseases (The Elsartan Case)

                        Prof. John Matsoukas(University of Patras, Greece)

10:20-10:40       The discovery of imidazo[4,5-b]pyridine derivatives as inhibitors of Aurora kinases

                        Dr. Vassilios Bavetsias(The Institute of Cancer Research, UK)

10:40-11:00      Polyfluoroketones: A Fascinating Tool in the Quest for iPLA2 Selective Inhibitors

                        Dr. Victoria Magrioti (University of Athens, Greece)

11:00-11:30       Coffee Break

 

 

4th Session

                        Chairs: Prof. Elias Couladouros (Agricultural University of Athens)

                                    Prof. Valentini Ragoussi (University of Athens)          

                                               

11:30-12:15      Natural And /Or Biologically Active Products: A Good Source Of Inspiration For The Development Of Methodologies

                        Prof. Janine Cossy (École Supérieure de Physique et de Chimie Industrelles ParisTech, France)

12:15-12:40       Aryliodonium Ylides of Hydroxyquinones: Synthetic Applications

                        Prof. Spyros Spyroudis  (Aristotle University of Thessaloniki, Greece)

12:40-13:00       Natural Products: Mine of Inspiration

                        Dr. Alexandros L. Zografos  (Aristotle University of Thessaloniki, Greece)

13:00-14:00       Lunch Break

14:00-15:30       Poster Session

                        Coffee Break

 

 

5th Session

                        Chairs: Prof. Athanassios Giannis (University of Leipzig, Germany)

                                    Assoc. Prof. Thomas Mavromoustakos (University of Athens)

                                   

15:30-16:15       Catalytic Asymmetric Synthesis via Combined Metal and  Enzyme Catalysis

                        Prof. Jan-Erling Backvall (University of Stockholm, Sweden)

16:15-16:35       S-Oxide Activated Mannich Reactions in Medicinal Chemistry Enantioselective Synthesis of Substituted β-Lactams

                        Assoc. Prof. Plato A. Magriotis (University of Patras, Greece)

16:35-16:55       Sulfur Containing Nitrogen Heterocycles via 1,3-Dipolar Cycloadditions

                        Assoc. Prof. Yiannis Elemes (University of Ioannina, Greece)

16:55-17:15      Bacillus Subtilis Esterase (Bs2) and its Mutant E188W/M193C: Attractive Tools for the Selective Removal of Carboxyl Protecting Groups

                        Dr. Efrosini Barbayianni (University of Athens, Greece)

17:15-17:35       Independent Synthesis of DNA Pyrimidine Base Open Lesions and Study of their Cyclization Reaction

                        Monica-Violetta Circu (University of Athens, Greece)

 

SATURDAY, OCTOBER 17, 2009

 

6th Session

                        Chairs: Prof. Haralambos Katerinopoulos (University of Crete)

                                    Prof. Dionissios Papaioannou (University of Patras)

                                               

 

09:15-10:00      Multivalent, cooperative catalysts: from aggregation colloids to dendrimers, and nanoparticles

                        Prof. Paolo Scrimin (University of Padova, Italy)

10:00-10:25       Supramolecular architectures with carbon-based nanostructured materials

                        Dr. Nikos Tagmatarchis (National Hellenic Research Foundation, Greece)

10:25-10:45       Ruthenium-Based Metathesis Catalysts Coordinated with Heterocyclic Carbene Ligands: Synthesis, Structure, and Catalytic Activity

                        Dr. Georgios C. Vougioukalakis (NCSR “Demokritos”, Greece)

10:45-11:15       Coffee Break

 

 

7th Session

                        Chairs: Prof. Alexandre Alexakis (University of Geneva, Switzerland)

                                    As. Prof. Thanassis Gimisis (University of Athens)

 

11:15-12:00       When Simplicity leads to Complexity

                        Prof. Ilan Marek (Technion - Israel Institute of Technology, Israel)

12:00-12:45       Synthesis of Novel Aromatic Architectures: Bowls, Gears, and Knots

                        Prof. Jay Siegel (University of Zurich, Switzerland)

 

12:45                Closing Remarks